Database | Drugs (IC50) | NAT1_low (N = 296) | NAT1_high (N = 296) | Fold change | P value |
---|---|---|---|---|---|
GDSC_V1 | Daporinad_1248 | 0.20 ± 0.72 | 0.08 ± 0.12 | 0.397303447 | 0.004357953 |
GDSC_V2 | Vincristine_1818 | 0.47 ± 0.91 | 0.20 ± 0.25 | 0.425308419 | 9.58337E-07 |
GDSC_V2 | Gemcitabine_1190 | 1.55 ± 2.62 | 0.68 ± 1.09 | 0.440790109 | 2.09078E-07 |
GDSC_V2 | Docetaxel_1819 | 0.29 ± 0.51 | 0.14 ± 0.20 | 0.472369513 | 1.56627E-06 |
GDSC_V2 | Vinblastine_1004 | 0.06 ± 0.10 | 0.03 ± 0.04 | 0.473404913 | 1.09105E-06 |
GDSC_V1 | Gemcitabine_135 | 0.18 ± 0.23 | 0.10 ± 0.16 | 0.547522731 | 6.26625E-07 |
GDSC_V2 | YK-4-279_1239 | 17.78 ± 19.09 | 9.76 ± 10.37 | 0.549208082 | 4.43499E-10 |
GDSC_V2 | Pevonedistat_1529 | 3.86 ± 5.34 | 2.12 ± 2.12 | 0.550279084 | 2.91587E-07 |
GDSC_V2 | Vinorelbine_2048 | 0.09 ± 0.13 | 0.05 ± 0.08 | 0.566325708 | 2.46423E-06 |
GDSC_V2 | KRAS (G12C) Inhibitor-12_1855 | 129.49 ± 110.22 | 74.12 ± 61.28 | 0.572363494 | 1.60819E-13 |
GDSC_V1 | PLK_6522_1451 | 0.15 ± 0.46 | 0.09 ± 0.09 | 0.578548545 | 0.016226363 |
GDSC_V2 | Cytarabine_1006 | 9.78 ± 8.68 | 5.85 ± 8.29 | 0.597889224 | 2.66787E-08 |
GDSC_V1 | ARRY-520_474 | 0.10 ± 0.10 | 0.06 ± 0.07 | 0.599251363 | 1.38231E-07 |
GDSC_V1 | Ispinesib Mesylate_208 | 0.22 ± 0.24 | 0.13 ± 0.11 | 0.608238084 | 1.83669E-08 |
GDSC_V1 | AZD4877_1409 | 0.04 ± 0.04 | 0.03 ± 0.02 | 0.610253366 | 2.61266E-09 |
GDSC_V2 | Docetaxel_1007 | 0.02 ± 0.02 | 0.01 ± 9.5e-3 | 0.613821245 | 2.25472E-10 |
GDSC_V2 | Mitoxantrone_1810 | 3.31 ± 3.03 | 2.05 ± 2.01 | 0.619296618 | 4.2026E-09 |
GDSC_V2 | AZD5438_1401 | 14.02 ± 14.25 | 8.71 ± 9.32 | 0.62121301 | 1.15855E-07 |
GDSC_V2 | Dinaciclib_1180 | 0.09 ± 0.25 | 0.06 ± 0.03 | 0.634598278 | 0.019359769 |
GDSC_V2 | Trametinib_1372 | 2.93 ± 3.19 | 1.86 ± 1.41 | 0.635035452 | 1.81855E-07 |
GDSC_V2 | 5-Fluorouracil_1073 | 195.90 ± 165.46 | 124.57 ± 195.72 | 0.635917282 | 2.1338E-06 |
GDSC_V2 | Dactinomycin_1811 | 0.13 ± 0.07 | 0.08 ± 0.05 | 0.641649302 | 2.19666E-16 |
GDSC_V2 | Irinotecan_1088 | 21.85 ± 19.37 | 14.02 ± 11.35 | 0.641771455 | 3.45048E-09 |
GDSC_V2 | Camptothecin_1003 | 0.15 ± 0.14 | 0.09 ± 0.08 | 0.641825954 | 3.95048E-08 |
GDSC_V2 | Eg5_9814_1712 | 0.08 ± 0.08 | 0.05 ± 0.06 | 0.648021519 | 4.93084E-07 |
GDSC_V2 | Teniposide_1809 | 2.89 ± 2.52 | 1.87 ± 1.68 | 0.648712054 | 1.35274E-08 |
GDSC_V2 | Alisertib_1051 | 11.96 ± 10.25 | 7.80 ± 7.41 | 0.651939165 | 2.3292E-08 |
GDSC_V2 | Paclitaxel_1080 | 0.11 ± 0.13 | 0.08 ± 0.13 | 0.655343737 | 0.000266396 |